L-822179

CAS No. 215874-86-5

L-822179 ( L 822179; L822179; L-822,179; L 822,179; L822,179 )

Catalog No. M27776 CAS No. 215874-86-5

L-822179 (α5IA) is a selective inverse agonist for the Α5 subtype of GABAA receptor with higher intrinsic activity at the A5 subtype than other drugs.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 115 In Stock
10MG 173 In Stock
25MG 293 In Stock
50MG 437 In Stock
100MG 626 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    L-822179
  • Note
    Research use only, not for human use.
  • Brief Description
    L-822179 (α5IA) is a selective inverse agonist for the Α5 subtype of GABAA receptor with higher intrinsic activity at the A5 subtype than other drugs.
  • Description
    L-822179 (α5IA) is a selective inverse agonist for the Α5 subtype of GABAA receptor with higher intrinsic activity at the A5 subtype than other drugs.
  • Synonyms
    L 822179; L822179; L-822,179; L 822,179; L822,179
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    MIF
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    215874-86-5
  • Formula Weight
    362.4
  • Molecular Formula
    C17H14N8O2
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    Cc1cc(no1)-c1nnc2c3ccccc3c(OCc3cn(C)nn3)nn12
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Zapatero MC, Pérez P, Vázquez MJ, Colmenarejo G, de Los Frailes M, Ramón F. Discovery of Novel Inhibitors of the Tautomerase Activity of Macrophage Migration Inhibitory Factor (MIF). J Biomol Screen. 2016 Jun;21(5):446-58.
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