KPT-6566 ( —— )

Catalog No. M20699 CAS No. 881487-77-0

KPT-6566 is a novel selective covalent pin1 inhibitor KPT-6566 shows an IC50 of 640?nM and a Ki of 625.2 nM for PIN1 PPIase domainand has anti-cancer activity.

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

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25MG	678	In Stock
50MG	954	In Stock
100MG	1287	In Stock
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Biological Information

Product Name

KPT-6566
Note

Research use only not for human use.
Brief Description

KPT-6566 is a novel selective covalent pin1 inhibitor KPT-6566 shows an IC50 of 640?nM and a Ki of 625.2 nM for PIN1 PPIase domainand has anti-cancer activity.
Description

KPT-6566 is a novel selective covalent pin1 inhibitor KPT-6566 shows an IC50 of 640?nM and a Ki of 625.2 nM for PIN1 PPIase domainand has anti-cancer activity.
Synonyms

——
Pathway

Others
Target

Other Targets
Recptor

PIN1 PPIase
Research Area

——
Indication

——

Chemical Information

CAS Number

881487-77-0
Formula Weight

443.5
Molecular Formula

C22H21NO5S2??
Purity

>98% (HPLC)
Solubility

DMSO:120 mg/mL?(270.55 mM)
SMILES

CC(C)(C)c1ccc(cc1)S(=O)(=O)\N=C1/C=C(SCC(O)=O)C(=O)c2ccccc12
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1.Zhang J Zhao F Yu X et al. Pharmacokinetics of eupalinolide A eupalinolide B and hyperoside from Eupatorium lindleyanum in rats by LC/MS/MS[J]. Journal of Chromatography B 2015 995-996:1-7.

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