JNJ-5207852
CAS No. 398473-34-2
JNJ-5207852 ( —— )
Catalog No. M20744 CAS No. 398473-34-2
JNJ-5207852 is a novel non-imidazole histamine H3 receptor antagonist with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
2MG | 40 | In Stock |
|
5MG | 65 | In Stock |
|
10MG | 102 | In Stock |
|
25MG | 215 | In Stock |
|
50MG | 426 | In Stock |
|
100MG | 624 | In Stock |
|
200MG | Get Quote | In Stock |
|
500MG | Get Quote | In Stock |
|
1G | Get Quote | In Stock |
|
Biological Information
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Product NameJNJ-5207852
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NoteResearch use only not for human use.
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Brief DescriptionJNJ-5207852 is a novel non-imidazole histamine H3 receptor antagonist with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor.
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DescriptionJNJ-5207852 is a novel non-imidazole histamine H3 receptor antagonist with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor.
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Synonyms——
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PathwayGPCR/G Protein
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TargetHistamine Receptor
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RecptorH3 receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number398473-34-2
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Formula Weight316.48
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Molecular FormulaC20H32N2O
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Purity>98% (HPLC)
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SolubilityDMSO:77.5 mg/mL (244.88 mM)
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SMILESC(COc1ccc(CN2CCCCC2)cc1)CN1CCCCC1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Esbenshade T A Browman K E Bitner R S et al. The histamine H3 receptor: an attractive target for the treatment of cognitive disorders[J]. 2008 154(6):1166-1181.
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