JNJ-31020028

CAS No. 1094873-14-9

JNJ-31020028 ( JNJ31020028; JNJ 31020028; JNJ-31020028 )

Catalog No. M10369 CAS No. 1094873-14-9

JNJ-31020028 is a selective brain penetrant antagonist of neuropeptide Y2 receptor with high affinity(pIC50=8.07, human; pIC50=8.22 rat).

Purity : >98%(HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 40 In Stock
5MG 65 In Stock
10MG 105 In Stock
25MG 194 In Stock
50MG 335 In Stock
100MG 500 In Stock
500MG 1098 In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    JNJ-31020028
  • Note
    Research use only, not for human use.
  • Brief Description
    JNJ-31020028 is a selective brain penetrant antagonist of neuropeptide Y2 receptor with high affinity(pIC50=8.07, human; pIC50=8.22 rat).
  • Description
    JNJ-31020028 is a selective brain penetrant antagonist of neuropeptide Y2 receptor with high affinity(pIC50=8.07, human; pIC50=8.22 rat); >100-fold selective versus human Y1/Y4/Y5 receptors.
  • Synonyms
    JNJ31020028; JNJ 31020028; JNJ-31020028
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    Y2 receptor
  • Research Area
    Neurological Disease
  • Indication
    ——

Chemical Information

  • CAS Number
    1094873-14-9
  • Formula Weight
    565.68
  • Molecular Formula
    C34H36FN5O2
  • Purity
    >98%(HPLC)
  • Solubility
    DMSO: 10 mM
  • SMILES
    O=C(NC1=CC=C(N2CCN(C(C3=CC=CC=C3)C(N(CC)CC)=O)CC2)C(F)=C1)C4=CC=CC=C4C5=CC=CN=C5
  • Chemical Name
    N-(4-(4-(2-(diethylamino)-2-oxo-1-phenylethyl)piperazin-1-yl)-3-fluorophenyl)-2-(pyridin-3-yl)benzamide

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Shoblock JR, et al. Psychopharmacology (Berl). 2010 Feb;208(2):265-77.
molnova catalog
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