IPI-3063

CAS No. 1425043-73-7

IPI-3063 ( —— )

Catalog No. M23579 CAS No. 1425043-73-7

IPI-3063 is an effective and selective inhibitor of PI3K p110δ (IC50: 2.5?±?1.2 nM).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 87 In Stock
5MG 160 In Stock
10MG 267 In Stock
25MG 537 In Stock
50MG 764 In Stock
100MG 1017 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    IPI-3063
  • Note
    Research use only, not for human use.
  • Brief Description
    IPI-3063 is an effective and selective inhibitor of PI3K p110δ (IC50: 2.5?±?1.2 nM).
  • Description
    IPI-3063 is an effective and selective inhibitor of PI3K p110δ (IC50: 2.5?±?1.2 nM).
  • Synonyms
    ——
  • Pathway
    PI3K/Akt/mTOR signaling
  • Target
    PI3K
  • Recptor
    p110α;p110β;p110γ;p110δ
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1425043-73-7
  • Formula Weight
    455.5
  • Molecular Formula
    C25H25N7O2
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:83.33 mg/mL (182.94 mM)
  • SMILES
    C[C@@H](C1=CC2=C(C(=CC=C2)C3=CN(C(=O)C=C3)C)C(=O)N1C(C)C)NC4=NC=NC(=C4C#N)N
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Chiu H, et al. The Selective Phosphoinoside-3-Kinase p110δ Inhibitor IPI-3063 Potently Suppresses B Cell Survival, Proliferation, and Differentiation. Front Immunol. 2017 Jun 30;8:747.
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