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Halopemide
CAS No. 59831-65-1
Halopemide( —— )
Catalog No. M26708 CAS No. 59831-65-1
Halopemide is a potent inhibitor of PLD (IC50 = 220 and 310 nM for human PLD1 and PLD2). Halopemid is an antagonist of dopamine receptors. Halopemid can be used in psychotropic research.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 115 | Get Quote |
|
| 10MG | 192 | Get Quote |
|
| 25MG | 385 | Get Quote |
|
| 50MG | 575 | Get Quote |
|
| 100MG | 801 | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameHalopemide
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NoteResearch use only, not for human use.
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Brief DescriptionHalopemide is a potent inhibitor of PLD (IC50 = 220 and 310 nM for human PLD1 and PLD2). Halopemid is an antagonist of dopamine receptors. Halopemid can be used in psychotropic research.
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DescriptionHalopemide is a potent inhibitor of PLD (IC50 = 220 and 310 nM for human PLD1 and PLD2). Halopemid is an antagonist of dopamine receptors. Halopemid can be used in psychotropic research.(In Vitro):In transdifferentiated MOVAS cells, Halopemide (1-2 μM; 21 days) influences calcification.(In Vivo):In the majority of monkeys tested, Halopemide (10 mg/kg; p.o.) causes dyskinesias.
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In VitroHalopemide (1-2 μM; 21 day) affects calcification in transdifferentiated MOVAS cells.
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In VivoHalopemide (10 mg/kg; p.o.) induces dyskinesias in the majority of monkeys tested.
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Synonyms——
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PathwayOthers
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TargetOther Targets
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RecptorCDK9
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Research Area——
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Indication——
Chemical Information
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CAS Number59831-65-1
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Formula Weight416.88
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Molecular FormulaC21H22ClFN4O2
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 41.67 mg/mL (99.96 mM)
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SMILESFc1ccc(cc1)C(=O)NCCN1CCC(CC1)n1c2ccc(Cl)cc2[nH]c1=O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Sabbah M, et al. Fragment-Based Design of Mycobacterium tuberculosis InhA Inhibitors. J Med Chem. 2020 May 14;63(9):4749-4761.
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