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Halopemide

CAS No. 59831-65-1

Halopemide( —— )

Catalog No. M26708 CAS No. 59831-65-1

Halopemide is a potent inhibitor of PLD (IC50 = 220 and 310 nM for human PLD1 and PLD2). Halopemid is an antagonist of dopamine receptors. Halopemid can be used in psychotropic research.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    Halopemide
  • Note
    Research use only, not for human use.
  • Brief Description
    Halopemide is a potent inhibitor of PLD (IC50 = 220 and 310 nM for human PLD1 and PLD2). Halopemid is an antagonist of dopamine receptors. Halopemid can be used in psychotropic research.
  • Description
    Halopemide is a potent inhibitor of PLD (IC50 = 220 and 310 nM for human PLD1 and PLD2). Halopemid is an antagonist of dopamine receptors. Halopemid can be used in psychotropic research.(In Vitro):In transdifferentiated MOVAS cells, Halopemide (1-2 μM; 21 days) influences calcification.(In Vivo):In the majority of monkeys tested, Halopemide (10 mg/kg; p.o.) causes dyskinesias.
  • In Vitro
    Halopemide (1-2 μM; 21 day) affects calcification in transdifferentiated MOVAS cells.
  • In Vivo
    Halopemide (10 mg/kg; p.o.) induces dyskinesias in the majority of monkeys tested.
  • Synonyms
    ——
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    CDK9
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    59831-65-1
  • Formula Weight
    416.88
  • Molecular Formula
    C21H22ClFN4O2
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 41.67 mg/mL (99.96 mM)
  • SMILES
    Fc1ccc(cc1)C(=O)NCCN1CCC(CC1)n1c2ccc(Cl)cc2[nH]c1=O
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Sabbah M, et al. Fragment-Based Design of Mycobacterium tuberculosis InhA Inhibitors. J Med Chem. 2020 May 14;63(9):4749-4761.
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