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Glutaminase-IN-3
CAS No. 1439399-45-7
Glutaminase-IN-3( —— )
Catalog No. M34941 CAS No. 1439399-45-7
Glutaminase-IN-3 is a potent Glutaminase 1 inhibitor with potential antitumor activity and inhibits GLS1 for cancer research.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 54 | Get Quote |
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| 10MG | 77 | Get Quote |
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| 25MG | 118 | Get Quote |
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| 50MG | 174 | Get Quote |
|
| 100MG | 251 | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameGlutaminase-IN-3
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NoteResearch use only, not for human use.
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Brief DescriptionGlutaminase-IN-3 is a potent Glutaminase 1 inhibitor with potential antitumor activity and inhibits GLS1 for cancer research.
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DescriptionGlutaminase-IN-3 (compound 657) is a potent glutaminase inhibitor with an IC50 of 0.24 μM for Glutaminase 1 (GLS1). Glutaminase-IN-3 is extracted from patent WO2014089048A1, compound 657.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayOthers
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TargetOther Targets
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RecptorGlutaminase
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Research Area——
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Indication——
Chemical Information
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CAS Number1439399-45-7
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Formula Weight452.45
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Molecular FormulaC19H19F3N6O2S
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 50 mg/mL (110.51 mM; Ultrasonic )
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SMILESFC(F)(F)Oc1cccc(CC(=O)N=c2ccc(CCCCc3n[nH]c(=N)s3)n[nH]2)c1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Mark K. Bennett, et al. Treatment of cancer with heterocyclic inhibitors of glutaminase. WO2014089048A1.
molnova catalog
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