GSK2830371
CAS No. 1404456-53-6
GSK2830371( GSK 2830371 | GSK2830371 | GSK-2830371 )
Catalog No. M17279 CAS No. 1404456-53-6
GSK2830371 is an orally active, allosteric Wip1 phosphatase inhibitor with IC50 of 6 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
5MG | 43 | In Stock |
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10MG | 74 | In Stock |
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25MG | 138 | In Stock |
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50MG | 240 | In Stock |
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100MG | 402 | In Stock |
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200MG | Get Quote | In Stock |
|
500MG | Get Quote | In Stock |
|
1G | Get Quote | In Stock |
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Biological Information
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Product NameGSK2830371
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NoteResearch use only, not for human use.
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Brief DescriptionGSK2830371 is an orally active, allosteric Wip1 phosphatase inhibitor with IC50 of 6 nM.
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DescriptionGSK 2830371 is a WiP1 inhibitor. It inhibits cell growth and tumor growth in lymphoma and neuroblastoma models.
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In Vitro——
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In Vivo——
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SynonymsGSK 2830371 | GSK2830371 | GSK-2830371
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PathwayAngiogenesis
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TargetFGFR
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RecptorWip1 phosphatase
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number1404456-53-6
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Formula Weight461.02
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Molecular FormulaC23H29ClN4O2S
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Purity>98% (HPLC)
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SolubilityDMSO : ≥ 51 mg/mL. 110.62 mM
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SMILESCC1=NC=C(Cl)C=C1NCC1=CC=C(S1)C(=O)N[C@@H](CC1CCCC1)C(=O)NC1CC1
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Chemical Name(S)-5-(((5-chloro-2-methylpyridin-3-yl)amino)methyl)-N-(3-cyclopentyl-1-(cyclopropylamino)-1-oxopropan-2-yl)thiophene-2-carboxamide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Gilmartin AG, et al. Nat Chem Biol. 2014, 10(3), 181-187
molnova catalog
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