GSK2830371

CAS No. 1404456-53-6

GSK2830371( GSK 2830371 | GSK2830371 | GSK-2830371 )

Catalog No. M17279 CAS No. 1404456-53-6

GSK2830371 is an orally active, allosteric Wip1 phosphatase inhibitor with IC50 of 6 nM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 43 In Stock
10MG 74 In Stock
25MG 138 In Stock
50MG 240 In Stock
100MG 402 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    GSK2830371
  • Note
    Research use only, not for human use.
  • Brief Description
    GSK2830371 is an orally active, allosteric Wip1 phosphatase inhibitor with IC50 of 6 nM.
  • Description
    GSK 2830371 is a WiP1 inhibitor. It inhibits cell growth and tumor growth in lymphoma and neuroblastoma models.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    GSK 2830371 | GSK2830371 | GSK-2830371
  • Pathway
    Angiogenesis
  • Target
    FGFR
  • Recptor
    Wip1 phosphatase
  • Research Area
    Cancer
  • Indication
    ——

Chemical Information

  • CAS Number
    1404456-53-6
  • Formula Weight
    461.02
  • Molecular Formula
    C23H29ClN4O2S
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO : ≥ 51 mg/mL. 110.62 mM
  • SMILES
    CC1=NC=C(Cl)C=C1NCC1=CC=C(S1)C(=O)N[C@@H](CC1CCCC1)C(=O)NC1CC1
  • Chemical Name
    (S)-5-(((5-chloro-2-methylpyridin-3-yl)amino)methyl)-N-(3-cyclopentyl-1-(cyclopropylamino)-1-oxopropan-2-yl)thiophene-2-carboxamide

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Gilmartin AG, et al. Nat Chem Biol. 2014, 10(3), 181-187
molnova catalog
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