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GSK137647A

CAS No. 349085-82-1

GSK137647A ( GSK137647A; GSK-137647A )

Catalog No. M17492 CAS No. 349085-82-1

GSK137647A is a selective FFA4 agonist.

Purity : 98%

COA

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HNMR

HPLC

MSDS

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Size	Price / USD	Stock	Quantity
2MG	27	In Stock
5MG	42	In Stock
10MG	69	In Stock
25MG	141	In Stock
50MG	231	In Stock
100MG	402	In Stock
200MG	581	In Stock
500MG	888	In Stock
1G	Get Quote	In Stock

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Biological Information

Product Name

GSK137647A
Note

Research use only, not for human use.
Brief Description

GSK137647A is a selective FFA4 agonist.
Description

GSK137647A is an agonist of the free fatty acid receptor 4 (FFA4/GPR120) with pEC50s = 6.3, 6.2, and 6.1 at human, mouse, and rat receptors, respectively. GSK137647A is selective for GPR120 over a panel of 61 other targets, including other FFARs.
Synonyms

GSK137647A; GSK-137647A
Pathway

Endocrinology/Hormones
Target

AChR
Recptor

GPR120
Research Area

Metabolic Disease
Indication

——

Chemical Information

CAS Number

349085-82-1
Formula Weight

305.39
Molecular Formula

C16H19NO3S
Purity

98%
Solubility

DMSO : ≥ 32 mg/mL. 104.78 mM; H2O : < 0.1 mg/mL
SMILES

Cc1cc(c(c(c1)C)NS(=O)(=O)c1ccc(cc1)OC)C
Chemical Name

4-methoxy-N-(2,4,6-trimethylphenyl)-benzenesulfonamide

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1. Sparks SM. Etal. Bioorg Med Chem Lett. 2014 Jul 15;24(14):3100-3.

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