GSK-239512

CAS No. 720691-69-0

GSK-239512 ( GSK239512; GSK 239512 )

Catalog No. M27879 CAS No. 720691-69-0

GSK-239512 is an antagonist of H3 receptor and can be used in studies about the treatment of cognitive dysfunction in neurodegenerative disorders.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 131 Get Quote
10MG 173 Get Quote
25MG 312 Get Quote
50MG 464 Get Quote
100MG 672 Get Quote
200MG Get Quote Get Quote
500MG Get Quote Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    GSK-239512
  • Note
    Research use only, not for human use.
  • Brief Description
    GSK-239512 is an antagonist of H3 receptor and can be used in studies about the treatment of cognitive dysfunction in neurodegenerative disorders.
  • Description
    GSK-239512 is an antagonist of H3 receptor and can be used in studies about the treatment of cognitive dysfunction in neurodegenerative disorders.
  • Synonyms
    GSK239512; GSK 239512
  • Pathway
    GPCR/G Protein
  • Target
    Histamine Receptor
  • Recptor
    5-HT2;D4 Receptor
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    720691-69-0
  • Formula Weight
    377.5
  • Molecular Formula
    C23H27N3O2
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    O=C1CCCN1c1ccc(Oc2ccc3CCN(CCc3c2)C2CCC2)nc1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Malgouris C, et al. Autoradiographic studies of RP 62203, a potent 5-HT2 receptor antagonist. In vitro and ex vivo selectivity profile. Eur J Pharmacol. 1993 Mar 16;233(1):29-35.
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