GLP-1R modulator L7-028

CAS No. 2648317-95-5

GLP-1R modulator L7-028( —— )

Catalog No. M35193 CAS No. 2648317-95-5

GLP-1R modulator L7-028 is a variant that enhances affinity for GLP-1 and (cAMP) signaling.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 132 In Stock
10MG 188 In Stock
25MG 322 In Stock
50MG 460 In Stock
100MG 684 In Stock
200MG 918 In Stock
500MG Get Quote In Stock
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Biological Information

  • Product Name
    GLP-1R modulator L7-028
  • Note
    Research use only, not for human use.
  • Brief Description
    GLP-1R modulator L7-028 is a variant that enhances affinity for GLP-1 and (cAMP) signaling.
  • Description
    GLP-1R modulator L7-028 is an allosteric modulator enhancing GLP-1 binding to GLP-1R via a transmembrane site (EC50 11.01 ± 2.73 μM).
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    GPCR/G Protein
  • Target
    Glucagon Receptor
  • Recptor
    Glucagon Receptor | cAMP
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2648317-95-5
  • Formula Weight
    392.49
  • Molecular Formula
    C24H28N2O3
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 100 mg/mL (254.78 mM; Ultrasonic )
  • SMILES
    O=C(Nc1cccc(c1)C(=O)N1CCCCC1)c1cccc(OC2CCCC2)c1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Wang J, et al. Allosteric Modulators Enhancing GLP-1 Binding to GLP-1R via a Transmembrane Site. ACS Chem Biol. 2021 Nov 19;16(11):2444-2452. ?
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