GCN2-IN-1

CAS No. 1448693-69-3

GCN2-IN-1 ( A-92 )

Catalog No. M26227 CAS No. 1448693-69-3

GCN2-IN-1 is an effective GCN2 inhibitor and can be used in research on the treatment of cancer as a chemotherapeutic agent.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 132 Get Quote
10MG 205 Get Quote
25MG 430 Get Quote
50MG 620 Get Quote
100MG 884 Get Quote
500MG 1764 Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    GCN2-IN-1
  • Note
    Research use only, not for human use.
  • Brief Description
    GCN2-IN-1 is an effective GCN2 inhibitor and can be used in research on the treatment of cancer as a chemotherapeutic agent.
  • Description
    GCN2-IN-1 is an effective GCN2 inhibitor and can be used in research on the treatment of cancer as a chemotherapeutic agent.(In Vitro):GCN2-IN-1 inhibits GCN2 with an IC50 of <0.3 μM in the enzyme assay and an IC50 of 0.3-3 μM in the cell assay.
  • Synonyms
    A-92
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    ATPase
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1448693-69-3
  • Formula Weight
    402.4
  • Molecular Formula
    C19H18N10O
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    C1CC(CCO1)n1cc(Nc2ncc3nnn(-c4ccc5cn[nH]c5c4)c3n2)cn1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Suga H, Asakura K, Sasaki S, Nojima M, Okubo H, Hirota N, Notsu A, Fukui M, Date C. Validation study of a self-administered diet history questionnaire for estimating amino acid intake among Japanese adults. Asia Pac J Clin Nutr. 2018;27(3):638-645.
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