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Flupirtine
CAS No. 56995-20-1
Flupirtine( D-9998 )
Catalog No. M15076 CAS No. 56995-20-1
A selective neuronal potassium channel (KCNQ/KV7 channel) activator that also has indirect NMDA receptor antagonist and GABAA receptor modulatory properties.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 873 | Get Quote |
|
| 50MG | 1782 | Get Quote |
|
| 100MG | 2250 | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameFlupirtine
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NoteResearch use only, not for human use.
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Brief DescriptionA selective neuronal potassium channel (KCNQ/KV7 channel) activator that also has indirect NMDA receptor antagonist and GABAA receptor modulatory properties.
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DescriptionA selective neuronal potassium channel (KCNQ/KV7 channel) activator that also has indirect NMDA receptor antagonist and GABAA receptor modulatory properties; a centrally acting non-opioid analgesic used as an analgesic for acute and chronic pain.Pain Discontinued.
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In Vitro——
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In Vivo——
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SynonymsD-9998
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PathwayCell Cycle/DNA Damage
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TargetPotassium Channel
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RecptorPotassium Channel
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Research AreaNeurological Disease
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IndicationPain
Chemical Information
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CAS Number56995-20-1
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Formula Weight304.3195
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Molecular FormulaC15H17FN4O2
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Purity>98% (HPLC)
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Solubility10 mM in DMSO
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SMILESCCOC(=O)NC1=C(N=C(C=C1)NCC2=CC=C(C=C2)F)N
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Chemical NameCarbamic acid, N-[2-amino-6-[[(4-fluorophenyl)methyl]amino]-3-pyridinyl]-, ethyl ester
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Szelenyi I, et al. Inflamm Res. 2013 Mar;62(3):251-8.
2. Harish S, et al. J Anaesthesiol Clin Pharmacol. 2012 Apr;28(2):172-7.
3. Hedegaard ER, et al. J Pharmacol Exp Ther. 2016 Apr;357(1):94-102.
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