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Entasobulin

CAS No. 501921-61-5

Entasobulin( —— )

Catalog No. M26678 CAS No. 501921-61-5

Entasobulin is an inhibitor of β-tubulin polymerization. It has a potential anticancer activity.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    Entasobulin
  • Note
    Research use only, not for human use.
  • Brief Description
    Entasobulin is an inhibitor of β-tubulin polymerization. It has a potential anticancer activity.
  • Description
    Entasobulin is an inhibitor of β-tubulin polymerization. It has a potential anticancer activity.(In Vitro):Entasobulin is an indolizine-glyoxylamide based small molecule. It shows substantial in vitro anti-proliferative activities against cancer cell lines, including multidrug resistance (MDR) phenotypes.
  • In Vitro
    Entasobulin is a indolizine-glyoxylamide based small molecule that demonstrate substantial in vitro anti-proliferative activities against cancer cell lines, including multidrug resistance (MDR) phenotypes.
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Cytoskeleton/Cell Adhesion Molecules
  • Target
    Microtubule/Tubulin
  • Recptor
    MLLT1| MLLT3
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    501921-61-5
  • Formula Weight
    439.9
  • Molecular Formula
    C26H18ClN3O2
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 155 mg/mL (352.36 mM)
  • SMILES
    Clc1ccc(Cn2cc(C(=O)C(=O)Nc3ccc4ncccc4c3)c3ccccc23)cc1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Moustakim M, et al. Discovery of an MLLT1/3 YEATS Domain Chemical Probe. Angew Chem Int Ed Engl. 2018 Dec 10;57(50):16302-16307.
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