Enpp-1-IN-16

CAS No. 2289739-47-3

Enpp-1-IN-16( —— )

Catalog No. M37145 CAS No. 2289739-47-3

Enpp-1-IN-16 is an inhibitor targeting ENPP1 with potential anti-cancer activity.Enpp-1-IN-16 can be used to study insulin resistance in relation to type II diabetes mellitus and various ENPP1-mediated diseases in the chondrocalcinosis and osteoarthritis classes.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 76 Get Quote
10MG 122 Get Quote
25MG 266 Get Quote
50MG 419 Get Quote
100MG 647 Get Quote
500MG 1341 Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    Enpp-1-IN-16
  • Note
    Research use only, not for human use.
  • Brief Description
    Enpp-1-IN-16 is an inhibitor targeting ENPP1 with potential anti-cancer activity.Enpp-1-IN-16 can be used to study insulin resistance in relation to type II diabetes mellitus and various ENPP1-mediated diseases in the chondrocalcinosis and osteoarthritis classes.
  • Description
    Enpp-1-IN-16 (compound 54) is an ENPP1 inhibitor. Enpp-1-IN-16 has the potential to study cancer, especially in cases of high ENPP1 expression or elevated cytoplasmic DNA levels. Enpp-1-IN-16 can also be used in other diseases mediated by ENPP1, such as bacterial or viral infections, insulin resistance and type II diabetes, chondrocalcinosis and osteoarthritis, calcium pyrophosphate deposition disorder (CPPD), low Phosphatase disease and soft tissue calcification disorders.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Angiogenesis
  • Target
    PDE
  • Recptor
    PDE
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2289739-47-3
  • Formula Weight
    428.52
  • Molecular Formula
    C23H32N4O4
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 2 mg/mL (4.67 mM; Ultrasonic )
  • SMILES
    O=C(OC(C)(C)C)N1CCC2(C1)CCN(C=3N=CN=C4C=C(OC)C(OC)=CC43)CC2
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Derek A Cogan, et al. Imino sulfanone inhibitors of enpp1. WO2021225969A1.
molnova catalog
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