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Enpp-1-IN-16

CAS No. 2289739-47-3

Enpp-1-IN-16( —— )

Catalog No. M37145 CAS No. 2289739-47-3

Enpp-1-IN-16 is an inhibitor targeting ENPP1 with potential anti-cancer activity.Enpp-1-IN-16 can be used to study insulin resistance in relation to type II diabetes mellitus and various ENPP1-mediated diseases in the chondrocalcinosis and osteoarthritis classes.

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

Size	Price / USD	Stock	Quantity
5MG	76	Get Quote
10MG	122	Get Quote
25MG	266	Get Quote
50MG	419	Get Quote
100MG	647	Get Quote
500MG	1341	Get Quote
1G	Get Quote	Get Quote

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Biological Information

Product Name

Enpp-1-IN-16
Note

Research use only, not for human use.
Brief Description

Enpp-1-IN-16 is an inhibitor targeting ENPP1 with potential anti-cancer activity.Enpp-1-IN-16 can be used to study insulin resistance in relation to type II diabetes mellitus and various ENPP1-mediated diseases in the chondrocalcinosis and osteoarthritis classes.
Description

Enpp-1-IN-16 (compound 54) is an ENPP1 inhibitor. Enpp-1-IN-16 has the potential to study cancer, especially in cases of high ENPP1 expression or elevated cytoplasmic DNA levels. Enpp-1-IN-16 can also be used in other diseases mediated by ENPP1, such as bacterial or viral infections, insulin resistance and type II diabetes, chondrocalcinosis and osteoarthritis, calcium pyrophosphate deposition disorder (CPPD), low Phosphatase disease and soft tissue calcification disorders.
In Vitro

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In Vivo

——
Synonyms

——
Pathway

Angiogenesis
Target

PDE
Recptor

PDE
Research Area

——
Indication

——

Chemical Information

CAS Number

2289739-47-3
Formula Weight

428.52
Molecular Formula

C23H32N4O4
Purity

>98% (HPLC)
Solubility

In Vitro:?DMSO : 2 mg/mL (4.67 mM; Ultrasonic )
SMILES

O=C(OC(C)(C)C)N1CCC2(C1)CCN(C=3N=CN=C4C=C(OC)C(OC)=CC43)CC2
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1. Derek A Cogan, et al. Imino sulfanone inhibitors of enpp1. WO2021225969A1.

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