Eltoprazine

CAS No. 98224-03-4

Eltoprazine ( DU-28853 )

Catalog No. M16892 CAS No. 98224-03-4

An antiaggressive agent that acts as an agonist at the 5-HT1A and 5-HT1B receptors and as an antagonist at the 5-HT2C receptor.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 873 Get Quote
50MG 1782 Get Quote
100MG 2250 Get Quote
200MG Get Quote Get Quote
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Biological Information

  • Product Name
    Eltoprazine
  • Note
    Research use only, not for human use.
  • Brief Description
    An antiaggressive agent that acts as an agonist at the 5-HT1A and 5-HT1B receptors and as an antagonist at the 5-HT2C receptor.
  • Description
    An antiaggressive agent that acts as an agonist at the 5-HT1A and 5-HT1B receptors and as an antagonist at the 5-HT2C receptor.Schizophrenia Phase 2 Clinical
  • Synonyms
    DU-28853
  • Pathway
    Endocrinology/Hormones
  • Target
    5-HT Receptor
  • Recptor
    5-HT Receptor
  • Research Area
    Neurological Disease
  • Indication
    Schizophrenia

Chemical Information

  • CAS Number
    98224-03-4
  • Formula Weight
    220.27
  • Molecular Formula
    C12H16N2O2
  • Purity
    >98% (HPLC)
  • Solubility
    10 mM in DMSO
  • SMILES
    C1CN(CCN1)C2=C3C(=CC=C2)OCCO3.Cl
  • Chemical Name
    Piperazine, 1-(2,3-dihydro-1,4-benzodioxin-5-yl)-

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Sijbesma H, et al. Eur J Pharmacol. 1990 Feb 20;177(1-2):55-66.
2. Jols M, et al. J Pharmacol Exp Ther. 1990 Apr;253(1):284-9.
3. Mos J, et al. Eur J Pharmacol. 1992 Mar 3;212(2-3):295-8.
molnova catalog
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