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EPZ004777
CAS No. 1338466-77-5
EPZ004777 ( EPZ004777; EPZ 004777 )
Catalog No. M11359 CAS No. 1338466-77-5
EPZ004777 is a potent, selectiveDOT1Linhibitor withIC50of 0.4 nM.
Purity : >98%(HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 68 | In Stock |
|
| 10MG | 110 | In Stock |
|
| 25MG | 222 | In Stock |
|
| 50MG | 340 | In Stock |
|
| 100MG | 502 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameEPZ004777
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NoteResearch use only, not for human use.
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Brief DescriptionEPZ004777 is a potent, selectiveDOT1Linhibitor withIC50of 0.4 nM.
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DescriptionEPZ004777 is a potent, selectiveDOT1Linhibitor withIC50of 0.4 nM.
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SynonymsEPZ004777; EPZ 004777
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PathwayChromatin/Epigenetic
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TargetHMTase
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RecptorDOT1L
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number1338466-77-5
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Formula Weight539.67
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Molecular FormulaC28H41N7O4
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Purity>98%(HPLC)
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SolubilityEthanol: 100 mg/mL (185.29 mM); DMSO: 100 mg/mL (185.29 mM)
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SMILESO=C(NC1=CC=C(C(C)(C)C)C=C1)NCCCN(C[C@H]2O[C@@H](N3C=CC4=C(N)N=CN=C43)[C@H](O)[C@@H]2O)C(C)C
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Chemical Name1-(3-((((2R,3S,4R,5R)-5-(4-amino-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-3,4-dihydroxytetrahydrofuran-2-yl)methyl)(isopropyl)amino)propyl)-3-(4-(tert-butyl)phenyl)urea
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Daigle SR, et al. Y Cell. 2011, 20(1), 53-65.
molnova catalog
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