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Droloxifene
CAS No. 82413-20-5
Droloxifene ( 3-Hydroxytamoxifen;FK-435 )
Catalog No. M16060 CAS No. 82413-20-5
A nonsteroidal selective estrogen receptor modulator (SERM) that shows 10- to 60-fold increased affinity for the estrogen receptor compared with Tamoxifen.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 177 | Get Quote |
|
| 10MG | 267 | Get Quote |
|
| 25MG | 464 | Get Quote |
|
| 50MG | 662 | Get Quote |
|
| 100MG | 888 | Get Quote |
|
| 500MG | 1782 | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameDroloxifene
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NoteResearch use only, not for human use.
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Brief DescriptionA nonsteroidal selective estrogen receptor modulator (SERM) that shows 10- to 60-fold increased affinity for the estrogen receptor compared with Tamoxifen.
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DescriptionA nonsteroidal selective estrogen receptor modulator (SERM) that shows 10- to 60-fold increased affinity for the estrogen receptor compared with Tamoxifen; has reduced partial estrogen agonistic activity.Breast Cancer Phase 2 Clinical
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Synonyms3-Hydroxytamoxifen;FK-435
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PathwayEndocrinology/Hormones
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TargetEstrogen Receptor/ERR
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RecptorEstrogen Receptor/ERR
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Research AreaCancer
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IndicationBreast Cancer
Chemical Information
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CAS Number82413-20-5
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Formula Weight387.52
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Molecular FormulaC26H29NO2
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Purity>98% (HPLC)
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Solubility——
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SMILESCCC(=C(C1=CC=C(C=C1)OCCN(C)C)C2=CC(=CC=C2)O)C3=CC=CC=C3
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Chemical Name(Z)-4-(1-(4-(2-aminoethoxy)phenyl)-2-phenylbut-1-en-1-yl)phenol
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Rauschning W, et al. Breast Cancer Res Treat. 1994;31(1):83-94.
2. Hasmann M, et al. Cancer Lett. 1994 Sep 15;84(2):101-16.
3. Leng Y, et al. Eur J Pharmacol. 2000 Dec 8;409(2):123-31.
2. Hasmann M, et al. Cancer Lett. 1994 Sep 15;84(2):101-16.
3. Leng Y, et al. Eur J Pharmacol. 2000 Dec 8;409(2):123-31.
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