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DprE1-IN-25
CAS No. 1615713-87-5
DprE1-IN-25 ( MDK3875; MDK-3875; MDK 3875; DprE1-IN-2; DprE1IN2 )
Catalog No. M12351 CAS No. 1615713-87-5
A potent, noncovalent DprE1 inhibitor with IC50 of 43 nM, shows activity against Mycobacterium tuberculosis (Mtb) in vitro with MIC of 0.39 uM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 53 | In Stock |
|
| 5MG | 87 | In Stock |
|
| 10MG | 132 | In Stock |
|
| 25MG | 259 | In Stock |
|
| 50MG | 384 | In Stock |
|
| 100MG | Get Quote | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameDprE1-IN-25
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NoteResearch use only, not for human use.
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Brief DescriptionA potent, noncovalent DprE1 inhibitor with IC50 of 43 nM, shows activity against Mycobacterium tuberculosis (Mtb) in vitro with MIC of 0.39 uM.
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DescriptionA potent, noncovalent DprE1 inhibitor with IC50 of 43 nM, shows activity against Mycobacterium tuberculosis (Mtb) in vitro with MIC of 0.39 uM.
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SynonymsMDK3875; MDK-3875; MDK 3875; DprE1-IN-2; DprE1IN2
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PathwayGPCR/G Protein
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TargetAntibacterial
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RecptorDprE
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number1615713-87-5
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Formula Weight368.43
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Molecular FormulaC19H24N6O2
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Purity>98% (HPLC)
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SolubilityDMSO: ≥ 33 mg/mL
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SMILESO=C(C1=CN(CC2=NC=NC(N(C)C)=C2C)C3=CC(C)=CN=C31)NCCO
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Chemical Name1H-Pyrrolo[3,2-b]pyridine-3-carboxamide, 1-[[6-(dimethylamino)-5-methyl-4-pyrimidinyl]methyl]-N-(2-hydroxyethyl)-6-methyl-
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Shirude PS, et al. J Med Chem. 2014 Jul 10;57(13):5728-37.
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