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Ddr1-In-1

CAS No. 1449685-96-4

Ddr1-In-1 ( —— )

Catalog No. M17304 CAS No. 1449685-96-4

DDR1-IN-1 is an effective and specificDDR1receptor tyrosine kinase inhibitor (IC50: 105 nM), about 3-fold selectivity over DDR2.

Purity : 98%

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

Size	Price / USD	Stock	Quantity
2MG	43	In Stock
5MG	69	In Stock
10MG	105	In Stock
25MG	162	In Stock
50MG	259	In Stock
100MG	405	In Stock
200MG	Get Quote	In Stock
500MG	Get Quote	In Stock
1G	Get Quote	In Stock

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Biological Information

Product Name

Ddr1-In-1
Note

Research use only, not for human use.
Brief Description

DDR1-IN-1 is an effective and specificDDR1receptor tyrosine kinase inhibitor (IC50: 105 nM), about 3-fold selectivity over DDR2.
Description

DDR1-IN-1 is an effective and specificDDR1receptor tyrosine kinase inhibitor (IC50: 105 nM), about 3-fold selectivity over DDR2.
Synonyms

——
Pathway

Cell Cycle/DNA Damage
Target

DNA/RNA Synthesis
Recptor

DDR1; DDR2
Research Area

Cancer
Indication

——

Chemical Information

CAS Number

1449685-96-4
Formula Weight

552.6
Molecular Formula

C30H31F3N4O3
Purity

98%
Solubility

DMSO : ≥ 41 mg/mL. 74.20 mM
SMILES

CCN1CCN(CC1)Cc1c(cc(cc1)C(=O)Nc1cc(c(cc1)C)Oc1cc2c(cc1)NC(=O)C2)C(F)(F)F
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1. Kim HG, et al. ACS Chem Biol. 2013, 8(10), 2145-2150.

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