DUN73423

CAS No. 2414373-42-3

DUN73423( —— )

Catalog No. M36296 CAS No. 2414373-42-3

DUN73423 (RET-IN-21) is a potent tyrosine kinase (RET) inhibitor with antitumour activity for the study of cancer.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 73 Get Quote
5MG 117 Get Quote
10MG 180 Get Quote
25MG 296 Get Quote
50MG 441 Get Quote
100MG 618 Get Quote
500MG 1251 Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    DUN73423
  • Note
    Research use only, not for human use.
  • Brief Description
    DUN73423 (RET-IN-21) is a potent tyrosine kinase (RET) inhibitor with antitumour activity for the study of cancer.
  • Description
    RET-IN-21 is an inhibitor of receptor tyrosine kinase (RET), with the IC50 of 4.4 μM, that has antitumor activity.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Tyrosine Kinase
  • Target
    c-RET
  • Recptor
    c-RET
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2414373-42-3
  • Formula Weight
    344.37
  • Molecular Formula
    C19H16N6O
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    N(CC=1C=CN=CC1)C2=NC3=C(C=NN3C=C2)C4=CC=C(C(N)=O)C=C4
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Rebecca Newton, et al. Discovery and Optimization of wt-RET/KDR-Selective Inhibitors of RETV804M Kinase. ACS Med. Chem. Lett. 2020, 11, 4, 497–505
molnova catalog
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