DS12881479

CAS No. 2373065-59-7

DS12881479( —— )

Catalog No. M35456 CAS No. 2373065-59-7

DS12881479 can be used in cancer research which is a potent and selective inhibitor of Mnk1(IC 50 =21 nM) .

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 154 Get Quote
5MG 244 Get Quote
10MG 368 Get Quote
25MG 640 Get Quote
50MG 861 Get Quote
100MG 1107 Get Quote
200MG 1512 Get Quote
500MG Get Quote Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    DS12881479
  • Note
    Research use only, not for human use.
  • Brief Description
    DS12881479 can be used in cancer research which is a potent and selective inhibitor of Mnk1(IC 50 =21 nM) .
  • Description
    DS12881479 is a potent and selective Mnk1 inhibitor with an IC50 value of 21 nM. DS12881479 can be used in cancer research.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    MAPK/ERK Signaling
  • Target
    MNK
  • Recptor
    MNK
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2373065-59-7
  • Formula Weight
    301.41
  • Molecular Formula
    C16H19N3OS
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 250 mg/mL (829.43 mM; Ultrasonic )
  • SMILES
    CN1CCC(CC1)C(=O)Nc1ncc(s1)-c1ccccc1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Yumi Matsui, et al. A novel inhibitor stabilizes the inactive conformation of MAPK-interacting kinase 1. Acta Crystallogr F Struct Biol Commun. 2018 Mar 1;74(Pt 3):156-160.?
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