CeMMEC2

CAS No. 902955-25-3

CeMMEC2 ( CeMMEC 2 )

Catalog No. M16491 CAS No. 902955-25-3

CeMMEC2 is a novel potent BRD4 inhibitor with IC50 of 0.9 uM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    CeMMEC2
  • Note
    Research use only, not for human use.
  • Brief Description
    CeMMEC2 is a novel potent BRD4 inhibitor with IC50 of 0.9 uM.
  • Description
    CeMMEC2 is a novel potent BRD4 inhibitor with IC50 of 0.9 uM, binds to both bromodomains of BRD4, comparably to (S)-JQ1.
  • Synonyms
    CeMMEC 2
  • Pathway
    Chromatin/Epigenetic
  • Target
    Bromodomain
  • Recptor
    Bromodomain
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    902955-25-3
  • Formula Weight
    257.34
  • Molecular Formula
    C14H19N5
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    CC1=NN=C2C=CC(NCCC3=CCCCC3)=NN21
  • Chemical Name
    N-[2-(cyclohex-1-en-1-yl)ethyl]-3-methyl[1,2,4]triazolo[4,3-b]pyridazin-6-amine

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Sdelci S, et al. Nat Chem Biol. 2016 Jul;12(7):504-10.
2. Blank, J. et al. WPO patent WO/2014/191894 (2014).
molnova catalog
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