Cbl-b-IN-1

CAS No. 2368841-84-1

Cbl-b-IN-1( —— )

Catalog No. M34938 CAS No. 2368841-84-1

Cbl-b-IN-1 is a potent Cbl-b inhibitor (IC50 <100 nM) with potential anticancer activity for the study of intestinal inflammation.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    Cbl-b-IN-1
  • Note
    Research use only, not for human use.
  • Brief Description
    Cbl-b-IN-1 is a potent Cbl-b inhibitor (IC50 <100 nM) with potential anticancer activity for the study of intestinal inflammation.
  • Description
    Cbl-b-IN-1 (example 519) is a Cbl-b inhibitor, extracted from patent WO2019148005A1, with an IC50 <100 nM.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    Others
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2368841-84-1
  • Formula Weight
    498.631
  • Molecular Formula
    C29H34N6O2
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 60 mg/mL (120.33 mM; Ultrasonic (<60°C)
  • SMILES
    Cn1cnnc1CC1(COC1)c1cccc(NC(=O)c2cc(CN3CCC4(CC4)C3)cc(n2)C2CC2)c1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. BARSANTI PAUL A (US), et al. INHIBITORS OF CBL-B AND METHODS OF USE THEREOF. WO/2019/148005A1.
molnova catalog
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