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Cariprazine

CAS No. 839712-12-8

Cariprazine ( RGH-188 )

Catalog No. M19163 CAS No. 839712-12-8

Cariprazine is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate affinity for the 5-HT1A receptor (Ki=2.6 nM).

Purity : 98%

COA Datasheet HNMR HPLC MSDS Handing Instructions
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5MG 99 In Stock
10MG 170 In Stock
25MG 300 In Stock
50MG 447 In Stock
100MG 624 In Stock
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Biological Information

  • Product Name
    Cariprazine
  • Note
    Research use only, not for human use.
  • Brief Description
    Cariprazine is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate affinity for the 5-HT1A receptor (Ki=2.6 nM).
  • Description
    Cariprazine is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate affinity for the 5-HT1A receptor (Ki=2.6 nM).
  • Synonyms
    RGH-188
  • Pathway
    Cytoskeleton/Cell Adhesion Molecules
  • Target
    Akt
  • Recptor
    D3;D2;5-HT1A
  • Research Area
    Neurological Disease
  • Indication
    ——

Chemical Information

  • CAS Number
    839712-12-8
  • Formula Weight
    427.41
  • Molecular Formula
    C21H32Cl2N4O
  • Purity
    98%
  • Solubility
    ——
  • SMILES
    CN(C)C(=O)N[C@H]1CC[C@H](CCN2CCN(CC2)c2cccc(Cl)c2Cl)CC1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Seneca N,et al.Occupancy of dopamine D and D and serotonin 5-HTA receptors by the novel antipsychotic drug candidate, cariprazine (RGH-188), in monkey brain measured using positron emission tomography. Psychopharmacology (Berl). 2011 Dec;218(3):579-87.
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