CPI-360
CAS No. 1802175-06-9
CPI-360( CPI-360 | CPI360 | CPI 360 )
Catalog No. M17382 CAS No. 1802175-06-9
CPI-360 is a potent, selective, and SAM-competitive EZH1 inhibitor with IC50 of 102.3 nM, >100-fold selectivity over other methyltransferases.
CPI-360 is a potent, selective, and SAM-competitive EZH1 inhibitor with IC50 of 102.3 nM, >100-fold selectivity over other methyltransferases.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
5MG | 158 | Get Quote |
|
10MG | 257 | Get Quote |
|
25MG | 430 | Get Quote |
|
50MG | 618 | Get Quote |
|
100MG | 898 | Get Quote |
|
200MG | Get Quote | Get Quote |
|
500MG | Get Quote | Get Quote |
|
1G | Get Quote | Get Quote |
|
Biological Information
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Product NameCPI-360
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NoteResearch use only, not for human use.
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Brief DescriptionCPI-360 is a potent, selective, and SAM-competitive EZH1 inhibitor with IC50 of 102.3 nM, >100-fold selectivity over other methyltransferases.
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DescriptionCPI-360 is a potent, selective,and SAM-competitive EZH1 inhibitor with IC50 of 102.3 nM
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In Vitro——
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In Vivo——
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SynonymsCPI-360 | CPI360 | CPI 360
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PathwayOthers
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TargetOther Targets
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RecptorEZH1
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number1802175-06-9
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Formula Weight437.53
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Molecular FormulaC25H31N3O4
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Purity>98% (HPLC)
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SolubilityDMSO : ≥ 48.9 mg/mL; 111.76 mM
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SMILESCOC1=C(CNC(=O)C2=C(C)N([C@H](C)C3CCOCC3)C3=C2C=CC=C3)C(=O)NC(C)=C1
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Chemical Name(R)-N-((4-methoxy-6-methyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-2-methyl-1-(1-(tetrahydro-2H-pyran-4-yl)ethyl)-1H-indole-3-carboxamide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
molnova catalog
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