CPI-360

CAS No. 1802175-06-9

CPI-360 ( CPI-360; CPI360; CPI 360 )

Catalog No. M17382 CAS No. 1802175-06-9

CPI-360 is a potent, selective, and SAM-competitive EZH1 inhibitor with IC50 of 102.3 nM, >100-fold selectivity over other methyltransferases.

Purity : 98%

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 158 Get Quote
10MG 257 Get Quote
25MG 430 Get Quote
50MG 618 Get Quote
100MG 898 Get Quote
200MG Get Quote Get Quote
500MG Get Quote Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    CPI-360
  • Note
    Research use only, not for human use.
  • Brief Description
    CPI-360 is a potent, selective, and SAM-competitive EZH1 inhibitor with IC50 of 102.3 nM, >100-fold selectivity over other methyltransferases.
  • Description
    CPI-360 is a potent, selective,and SAM-competitive EZH1 inhibitor with IC50 of 102.3 nM
  • Synonyms
    CPI-360; CPI360; CPI 360
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    EZH1
  • Research Area
    Cancer
  • Indication
    ——

Chemical Information

  • CAS Number
    1802175-06-9
  • Formula Weight
    437.53
  • Molecular Formula
    C25H31N3O4
  • Purity
    98%
  • Solubility
    DMSO : ≥ 48.9 mg/mL; 111.76 mM
  • SMILES
    COC1=C(CNC(=O)C2=C(C)N([C@H](C)C3CCOCC3)C3=C2C=CC=C3)C(=O)NC(C)=C1
  • Chemical Name
    (R)-N-((4-methoxy-6-methyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-2-methyl-1-(1-(tetrahydro-2H-pyran-4-yl)ethyl)-1H-indole-3-carboxamide

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

molnova catalog
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