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Home - Products - Membrane Transporter/Ion Channel - Sodium Channel - CNV1014802

CNV1014802

CAS No. 934240-30-9

CNV1014802 ( GSK-1014802;CNV-1014802;Raxatrigine;Vixotrigine;BIIB074 )

Catalog No. M16676 CAS No. 934240-30-9

CNV1014802 (GSK-1014802, Raxatrigine, Vixotrigine, BIIB074) is a potent, selective Nav1.7 sodium channel blocker.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    CNV1014802
  • Note
    Research use only, not for human use.
  • Brief Description
    CNV1014802 (GSK-1014802, Raxatrigine, Vixotrigine, BIIB074) is a potent, selective Nav1.7 sodium channel blocker.
  • Description
    CNV1014802 (GSK-1014802, Raxatrigine, Vixotrigine, BIIB074) is a potent, selective Nav1.7 sodium channel blocker, shows analgesic effects and potential in the treatment of cognitive symptoms of schizophrenia in vivo. Pain Phase 2 Clinical
  • Synonyms
    GSK-1014802;CNV-1014802;Raxatrigine;Vixotrigine;BIIB074
  • Pathway
    Membrane Transporter/Ion Channel
  • Target
    Sodium Channel
  • Recptor
    SodiumChannel
  • Research Area
    Neurological Disease
  • Indication
    Pain

Chemical Information

  • CAS Number
    934240-30-9
  • Formula Weight
    314.35
  • Molecular Formula
    C18H19FN2O2
  • Purity
    >98% (HPLC)
  • Solubility
    10 mM in DMSO
  • SMILES
    C1CC(NC1C2=CC=C(C=C2)OCC3=CC=CC=C3F)C(=O)N
  • Chemical Name
    2-Pyrrolidinecarboxamide, 5-[4-[(2-fluorophenyl)methoxy]phenyl]-, (2S,5R)-

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Bagal SK, et al. Bioorg Med Chem Lett. 2014 Aug 15;24(16):3690-9.
2. Deuis JR, et al. Toxins (Basel). 2016 Mar 17;8(3). pii: E78.
3. Zakrzewska JM, et al. Lancet Neurol. 2017 Apr;16(4):291-300.
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