CID3528206

CAS No. 674359-78-5

CID3528206( CID 3528206 )

Catalog No. M15572 CAS No. 674359-78-5

CID3528206 is a potent, small molecule yeast TORC1 inhibitor that inhibits TORC1 activity both in vitro and in vivo with IC50 of 150 nM and 3.9 uM, respectively.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    CID3528206
  • Note
    Research use only, not for human use.
  • Brief Description
    CID3528206 is a potent, small molecule yeast TORC1 inhibitor that inhibits TORC1 activity both in vitro and in vivo with IC50 of 150 nM and 3.9 uM, respectively.
  • Description
    CID3528206 is a potent, small molecule yeast TORC1 inhibitor that inhibits TORC1 activity both in vitro and in vivo with IC50 of 150 nM and 3.9 uM, respectively; alters GFP expression in all five GFP clones in a manner analogous to that of rapamycin, inhibits yeast cell growth.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    CID 3528206
  • Pathway
    PI3K/Akt/mTOR signaling
  • Target
    mTOR
  • Recptor
    mTOR
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    674359-78-5
  • Formula Weight
    278.247
  • Molecular Formula
    C11H11FN6O2
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    CNC1=NC(=C(C(=N1)NC2=CC(=CC=C2)F)[N+](=O)[O-])N
  • Chemical Name
    N4-(3-fluorophenyl)-N2-methyl-5-nitropyrimidine-2,4,6-triamine

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Chen J, et al. ACS Chem Biol. 2012 Apr 20;7(4):715-22.
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