Brexpiprazole

CAS No. 913611-97-9

Brexpiprazole( OPC 34712 )

Catalog No. M16564 CAS No. 913611-97-9

Brexpiprazole is a novel D2 dopamine partial agonist.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 41 In Stock
10MG 55 In Stock
25MG 66 In Stock
50MG 77 In Stock
100MG 91 In Stock
200MG 135 In Stock
500MG 259 In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Brexpiprazole
  • Note
    Research use only, not for human use.
  • Brief Description
    Brexpiprazole is a novel D2 dopamine partial agonist.
  • Description
    Brexpiprazole is a novel D2 dopamine partial agonist.
  • In Vitro
    ——
  • In Vivo
    Animal Model:Male C57BL/6NCrSlc mice, Dizocilpine (0.1 mg/kg) (HY-15084B) induced social recognition deficits Dosage:0.01, 0.03 and 0.1 mg/kg Administration:Oral administration, once Result:Significantly ameliorated Dizocilpine-induced social recognition deficits, without sedation or a reduction of exploratory behavior.
  • Synonyms
    OPC 34712
  • Pathway
    Endocrinology/Hormones
  • Target
    5-HT Receptor
  • Recptor
    5-HT1A| 5-HT2A| α1B-adrenergic receptor| α2C receptors| D2L
  • Research Area
    Neurological Disease
  • Indication
    ——

Chemical Information

  • CAS Number
    913611-97-9
  • Formula Weight
    433.57
  • Molecular Formula
    C25H27N3O2S
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO: 10 mM
  • SMILES
    O=C1NC2=C(C=C1)C=CC(OCCCCN1CCN(CC1)C1=C3C=CSC3=CC=C1)=C2
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Zajdel P, et al. Future Med Chem, 2014. 6(1): p. 57-75.
molnova catalog
related products
  • Ritanserin

    Ritanserin is a highly effective, relatively selective, long-acting antagonist of 5-HT2 receptor (IC50: 0.9 nM), less active on Histamine H1, Dopamine D2, Adrenergic α1, Adrenergic α2 receptors.

  • Vidofludimus

    Vidofludimus (4SC-101, SC12267) is a novel small molecule inhibitor of dihydroorotate dehydrogenase (DHODH).

  • 5-HT3 antagonist 3

    5-HT3 antagonist 3 (Compound 15b) is a high-affinity 5-HT3 receptor antagonist.