Bilastine

CAS No. 202189-78-4

Bilastine( Bilastine trade name Bilaxten )

Catalog No. M18206 CAS No. 202189-78-4

Bilastine is a novel new-generation antihistamine that is highly selective for the H1 histamine receptor, has a rapid onset and prolonged duration of action.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
25MG 35 In Stock
50MG 58 In Stock
100MG 95 In Stock
200MG 140 In Stock
500MG 236 In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Bilastine
  • Note
    Research use only, not for human use.
  • Brief Description
    Bilastine is a novel new-generation antihistamine that is highly selective for the H1 histamine receptor, has a rapid onset and prolonged duration of action.
  • Description
    Bilastine (trade name Bilaxten) is a second generation antihistamine drug for the treatment of allergic rhinoconjunctivitis and urticaria (hives). It exerts its effect as a selective histamine H1 receptor antagonist, and has a potency similar to cetirizine and is superior to fexofenadine. It was developed in Spain by FAES Farma. Bilastine is approved in the European Union for the symptomatic treatment of allergic rhinoconjunctivitis and urticaria, but it is not approved by the U.S. Food and Drug Administration for any use in the United States. Bilastine has been effective in the treatment of ocular symptoms and diseases of allergies, including rhinoconjuctivitis. Additionally, bilastine has been shown to improve quality of life, and all nasal and ocular symptoms related to allergic rhinitis.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    Bilastine trade name Bilaxten
  • Pathway
    Endocrinology/Hormones
  • Target
    5-HT Receptor
  • Recptor
    H1 receptor
  • Research Area
    Inflammation/Immunology
  • Indication
    ——

Chemical Information

  • CAS Number
    202189-78-4
  • Formula Weight
    463.62
  • Molecular Formula
    C28H37N3O3
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO : ≥ 49.3 mg/mL; 106.34 mM
  • SMILES
    CCOCCn1c(nc2ccccc12)C1CCN(CCc2ccc(cc2)C(C)(C)C(O)=O)CC1
  • Chemical Name
    2-(4-(2-(4-(1-(2-ethoxyethyl)-1H-benzo[d]imidazol-2-yl)piperidin-1-yl)ethyl)phenyl)-2-methylpropanoic acid

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Wolthers OD.Bilastine: a new nonsedating oral H1 antihistamine for treatment of allergic rhinoconjunctivitis and urticaria.Biomed Res Int. 2013;2013:626837.
molnova catalog
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