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BPTU
CAS No. 870544-59-5
BPTU ( BPTU; BMS-646786; BMS 646786 )
Catalog No. M17632 CAS No. 870544-59-5
Allosteric antagonist of P2Y1 (EC50 = 0.06-0.3 μM). Non-nucleotide ligand. Binds receptor outside of the helical bundle.
Purity : 98%
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 41 | In Stock |
|
| 5MG | 59 | In Stock |
|
| 10MG | 106 | In Stock |
|
| 25MG | 226 | In Stock |
|
| 50MG | 390 | In Stock |
|
| 100MG | 578 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameBPTU
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NoteResearch use only, not for human use.
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Brief DescriptionAllosteric antagonist of P2Y1 (EC50 = 0.06-0.3 μM). Non-nucleotide ligand. Binds receptor outside of the helical bundle.
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DescriptionAllosteric antagonist of P2Y1 (EC50 = 0.06-0.3 μM). Non-nucleotide ligand. Binds receptor outside of the helical bundle. Blocks inhibition of spontaneous contraction of rat and mouse colon induced by electrical field stimulation, nicotine and P2Y agonists. Antithrombotic; reduces platelet aggregation.
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SynonymsBPTU; BMS-646786; BMS 646786
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PathwayOthers
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TargetOther Targets
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RecptorP2Y1
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Research AreaCardiovascular Disease
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Indication——
Chemical Information
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CAS Number870544-59-5
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Formula Weight445.42
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Molecular FormulaC23H22F3N3O3
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Purity98%
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SolubilityDMSO : ≥ 33.3 mg/mL. 74.76 mM; H2O : < 0.1 mg/mL
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SMILESCC(C)(C)C1=CC=CC=C1OC2=C(C=CC=N2)NC(=O)NC3=CC=C(C=C3)OC(F)(F)F
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Chemical Name1-[2-(2-tert-Butylphenoxy)pyridin-3-yl]-3-[4-(trifluoromethoxy)phenyl]urea
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Abrahamsen B, et al. J Neurosci. 2013 Jan 16;33(3):1068-87.
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