BPDBA( —— )

Catalog No. M34193 CAS No. 312281-74-6

BPDBA is an effective, selective, and non-competitive inhibitor of the betaine/GABA transporter (BGT-1), displaying inhibitory activity against human BGT-1 and mouse GAT2, with IC50 values of 20 μM and 35 μM, respectively.

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

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10MG	85	Get Quote
25MG	170	Get Quote
50MG	273	Get Quote
100MG	431	Get Quote
500MG	945	Get Quote
1G	1251	Get Quote

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Biological Information

Product Name

BPDBA
Note

Research use only, not for human use.
Brief Description

BPDBA is an effective, selective, and non-competitive inhibitor of the betaine/GABA transporter (BGT-1), displaying inhibitory activity against human BGT-1 and mouse GAT2, with IC50 values of 20 μM and 35 μM, respectively.
Description

BPDBA is a selective and noncompetitive betaine/GABA transporter (BGT-1) inhibitor with IC50s of 20 μM and 35 μM against human BGT-1 and mouse GAT2, respectively.
In Vitro

——
In Vivo

——
Synonyms

——
Pathway

Others
Target

Other Targets
Recptor

GABA Receptor
Research Area

——
Indication

——

Chemical Information

CAS Number

312281-74-6
Formula Weight

363.28
Molecular Formula

C19H20Cl2N2O
Purity

>98% (HPLC)
Solubility

In Vitro:?DMSO : 100 mg/mL (275.27 mM; Ultrasonic )
SMILES

C(N1CCC(NC(=O)C2=C(Cl)C=C(Cl)C=C2)CC1)C3=CC=CC=C3
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1. Kragholm B, et al. Discovery of a subtype selective inhibitor of the human betaine/GABA transporter 1 (BGT-1) with a non-competitive pharmacological profile. Biochem Pharmacol. 2013 Aug 15;86(4):521-8.?

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