BML-277

CAS No. 516480-79-8

BML-277( BML-277 | C 3742 | Checkpoint Kinase 2 Inhibitor II )

Catalog No. M14798 CAS No. 516480-79-8

BML-277 (C 3742) is a selective Chk2 (checkpoint kinase 2) inhibitor with an IC50 of 15 nM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 42 In Stock
10MG 69 In Stock
25MG 143 In Stock
50MG 285 In Stock
100MG 426 In Stock
500MG 888 In Stock
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Biological Information

  • Product Name
    BML-277
  • Note
    Research use only, not for human use.
  • Brief Description
    BML-277 (C 3742) is a selective Chk2 (checkpoint kinase 2) inhibitor with an IC50 of 15 nM.
  • Description
    BML-277 (C 3742) is a selective Chk2 (checkpoint kinase 2) inhibitor with an IC50 of 15 nM.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    BML-277 | C 3742 | Checkpoint Kinase 2 Inhibitor II
  • Pathway
    Angiogenesis
  • Target
    Chk
  • Recptor
    Chk2
  • Research Area
    Cancer
  • Indication
    ——

Chemical Information

  • CAS Number
    516480-79-8
  • Formula Weight
    363.8
  • Molecular Formula
    C20H14ClN3O2
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO: 10 mM
  • SMILES
    O=C(C1=CC=C2C(N=C(C3=CC=C(OC4=CC=C(Cl)C=C4)C=C3)N2)=C1)N
  • Chemical Name
    2-(4-(4-Chlorophenoxy)phenyl)-1H-benzimidazole-5-carboxamide

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Arienti KL, et al. J Med Chem. 2005 Mar 24; 48(6): 1873-85.
molnova catalog
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