BGC201531

CAS No. 1186532-61-5

BGC201531( GTPL3380 | AP-1531 | BGC-20-1531 )

Catalog No. M23357 CAS No. 1186532-61-5

BGC201531 is a EP4 antagonist for the treatment of acute migraine.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 272 In Stock
10MG 408 In Stock
25MG 735 In Stock
100MG Get Quote In Stock
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Biological Information

  • Product Name
    BGC201531
  • Note
    Research use only, not for human use.
  • Brief Description
    BGC201531 is a EP4 antagonist for the treatment of acute migraine.
  • Description
    BGC201531 is a EP4 antagonist for the treatment of acute migraine.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    GTPL3380 | AP-1531 | BGC-20-1531
  • Pathway
    GPCR/G Protein
  • Target
    Prostaglandin Receptor
  • Recptor
    EP4
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1186532-61-5
  • Formula Weight
    496.58
  • Molecular Formula
    C26H28N2O6S
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    CC1=CC=CC=C1S(=O)(=O)[N-]C(=O)C2=CC(=C(O2)C)COC3=CC=C(C=C3)C4=NC=C(C=C4)OC.[Na+]
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Czigler A , Toth L , Szarka N , et al. Prostaglandin E2, a postulated mediator of neurovascular coupling, at low concentrations dilates whereas at higher concentrations constricts human cerebral parenchymal arterioles[J]. Prostaglandins & other lipid mediators, 2019, 146:106389.
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