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Azaphen dihydrochloride monohydrate

CAS No. 63302-99-8

Azaphen dihydrochloride monohydrate( —— )

Catalog No. M35587 CAS No. 63302-99-8

Azaphen dihydrochloride monohydrate (Pipofezin dihydrochloride monohydrate) is a serotonin reuptake inhibitor with antidepressant activity and sedative effects, which can be used to study neurological diseases.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
10MG 35 In Stock
25MG 54 In Stock
50MG 79 In Stock
100MG 113 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Azaphen dihydrochloride monohydrate
  • Note
    Research use only, not for human use.
  • Brief Description
    Azaphen dihydrochloride monohydrate (Pipofezin dihydrochloride monohydrate) is a serotonin reuptake inhibitor with antidepressant activity and sedative effects, which can be used to study neurological diseases.
  • Description
    Pipofezine(Azafen or Azaphen) is a potent inhibitor of the reuptake of serotonin. IC50 Value: Target: SSRIs Pipofezine is a tricyclic antidepressant (TCA) approved in Russia for the treatment ofdepression.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    GPCR/G Protein
  • Target
    5-HT Receptor
  • Recptor
    5-HT Receptor
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    63302-99-8
  • Formula Weight
    388.29
  • Molecular Formula
    C16H23Cl2N5O2
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?H2O : ≥ 100 mg/mL (257.54 mM) DMSO : 1 mg/mL (2.58 mM; Ultrasonic )
  • SMILES
    CN1C2=C(C=CC=C2)OC3=NN=C(N4CCN(CC4)C)C=C31.Cl.O.Cl
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Shinaev NN, Akzhigitov RG.Azaphen: a return to clinical practice.Zh Nevrol Psikhiatr Im S S Korsakova. 2005;105(10):55-6.?
molnova catalog
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