Apatinib

CAS No. 811803-05-1

Apatinib( YN968D1 )

Catalog No. M16035 CAS No. 811803-05-1

Apatinib is an orally bioavailable, selective VEGFR2 inhibitor with IC50 of 1 nM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 76 In Stock
5MG 108 In Stock
10MG 137 In Stock
25MG 233 In Stock
50MG 350 In Stock
100MG Get Quote In Stock
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Biological Information

  • Product Name
    Apatinib
  • Note
    Research use only, not for human use.
  • Brief Description
    Apatinib is an orally bioavailable, selective VEGFR2 inhibitor with IC50 of 1 nM.
  • Description
    Apatinib is an orally bioavailable, selective VEGFR2 inhibitor with IC50 of 1 nM.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    YN968D1
  • Pathway
    Angiogenesis
  • Target
    c-Kit
  • Recptor
    c-Kit| RET| c-Src| VEGFR2
  • Research Area
    Cancer
  • Indication
    ——

Chemical Information

  • CAS Number
    811803-05-1
  • Formula Weight
    397.48
  • Molecular Formula
    C24H23N5O
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO: 22 mg/mL (44.57 mM)
  • SMILES
    CS(O)(=O)=O.O=C(NC1=CC=C(C=C1)C1(CCCC1)C#N)C1=C(NCC2=CC=NC=C2)N=CC=C1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Tian S, et al. Y Sci, 2011, 102(7), 1374-1380.
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