Cart
sales@molnova.com
Abarelix
CAS No. 183552-38-7
Abarelix ( R3827; PPI 149 )
Catalog No. M23834 CAS No. 183552-38-7
Abarelix is a potent gonadotrophin-releasing hormone (GnRH) antagonist, which is used for prostate cancer treatment.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 79 | In Stock |
|
| 5MG | 122 | In Stock |
|
| 10MG | 201 | In Stock |
|
| 25MG | 438 | In Stock |
|
| 50MG | 626 | In Stock |
|
| 100MG | 888 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
-
Product NameAbarelix
-
NoteResearch use only, not for human use.
-
Brief DescriptionAbarelix is a potent gonadotrophin-releasing hormone (GnRH) antagonist, which is used for prostate cancer treatment.
-
DescriptionAbarelix is a potent gonadotrophin-releasing hormone (GnRH) antagonist, which is used for prostate cancer treatment.
-
SynonymsR3827; PPI 149
-
PathwayOthers
-
TargetOther Targets
-
RecptorGnRHR
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number183552-38-7
-
Formula Weight1416.1
-
Molecular FormulaC72H95ClN14O14
-
Purity>98% (HPLC)
-
SolubilityDMSO:14.2 mg/mL (10.03 mM)
-
SMILESC[C@H](C(=O)N)NC(=O)[C@@H]1CCCN1C(=O)[C@H](CCCCNC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](CC(=O)N)NC(=O)[C@H](CC2=CC=C(C=C2)O)N(C)C(=O)[C@H](CO)NC(=O)[C@@H](CC3=CN=CC=C3)NC(=O)[C@@H](CC4=CC=C(C=C4)Cl)NC(=O)[C@@H](CC5=CC6=CC=CC=C6C=C5)NC(=O)C
-
Chemical Name——
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1.Koechling W, et al. A novel GnRH antagonist, causes minimal histamine release compared with abarelix in an ex vivo model of human skin samples. Br J Clin Pharmacol. 2010 Oct;70(4):580-7.
molnova catalog
related products
-
Methyl 3-bromo-4,5-d...
Methyl 3-bromo-4,5-dihydroxybenzoate is a marine derived natural products found in Rhodomela confervoides.
-
Levothyroxine sodium
Levothyroxine, the major hormone derived from the thyroid gland, is the agonist of Thyroid hormone receptor alpha and beta.evothyroxine (L-T(4))can upregulate the expression of P-gp mRNA and protein in LS180 cells, but only L-T(4) and L-T(3) can produce the same effect in Caco-2 cells, which are relatively lacking in PXR.
-
3-Methoxytyramine
3-Methoxytyramine a well known extracellular metabolite of 3-hydroxytyramine/dopamine is a neuromodulator.
