AZ13705339 ( AZ-13705339; AZ 13705339 )

Catalog No. M27853 CAS No. 2016806-57-6

AZ13705339 is a potent and selective PAK1 inhibitor with IC50 of 0.33 nM.

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

Size	Price / USD	Stock	Quantity
2MG	35	Get Quote
5MG	58	Get Quote
10MG	88	Get Quote
25MG	200	Get Quote
50MG	320	Get Quote
100MG	515	Get Quote
200MG	Get Quote	Get Quote
500MG	Get Quote	Get Quote
1G	Get Quote	Get Quote

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Biological Information

Product Name

AZ13705339
Note

Research use only, not for human use.
Brief Description

AZ13705339 is a potent and selective PAK1 inhibitor with IC50 of 0.33 nM.
Description

AZ13705339 is a potent and selective PAK1 inhibitor with IC50 of 0.33 nM.(In Vitro):AZ13705339 (300 nM) prevents Siglec-8 binding-induced eosinophil death. In Namalwa cells, AZ13705339 (1 μM) inhibits αIgM-controlled but not PMA-induced adhesion.(In Vivo):In rats, AZ13705339 (100 mg/kg, p.o.) exhibits moderate clearance and Cmax of 7.7 μM.
Synonyms

AZ-13705339; AZ 13705339
Pathway

Others
Target

Other Targets
Recptor

——
Research Area

——
Indication

——

Chemical Information

CAS Number

2016806-57-6
Formula Weight

629.8
Molecular Formula

C33H36FN7O3S
Purity

>98% (HPLC)
Solubility

——
SMILES

CCS(=O)(=O)c1cc(Nc2ncc(F)c(n2)N(Cc2ccccc2C#N)c2cc(CO)ccc2C)ccc1N1CCN(C)CC1
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1.Andrew F Ducruet , et al. GM1485, a Nonimmunosuppressive Immunophilin Ligand, Promotes Neurofunctional Improvement and Neural Regeneration Following Stroke. J Neurosci Res. 2012 Jul;90(7):1413-23.

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