ASTX029

CAS No. 2095719-92-7

ASTX029 ( ASTX-029 )

Catalog No. M22011 CAS No. 2095719-92-7

ASTX029 is a selective and orally bioavailable extracellular signal-regulated kinases 1 and 2 (ERK 1/2) inhibitor, with potential antineoplastic activity.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 87 In Stock
10MG 140 In Stock
25MG 222 In Stock
50MG 402 In Stock
100MG 593 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    ASTX029
  • Note
    Research use only, not for human use.
  • Brief Description
    ASTX029 is a selective and orally bioavailable extracellular signal-regulated kinases 1 and 2 (ERK 1/2) inhibitor, with potential antineoplastic activity.
  • Description
    ASTX029 is a selective and orally bioavailable extracellular signal-regulated kinases 1 and 2 (ERK 1/2) inhibitor, with potential antineoplastic activity.
  • Synonyms
    ASTX-029
  • Pathway
    MAPK/ERK Signaling
  • Target
    ERK
  • Recptor
    ERK1/2
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2095719-92-7
  • Formula Weight
    584.04
  • Molecular Formula
    C29H31ClFN5O5
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:98 mg/mL (167.8 mM); Ethanol:48 mg/mL (82.2 mM)
  • SMILES
    COC1=CC(F)=CC(=C1)[C@@H](CO)NC(=O)[C@@H](C)N1CC2=CC=C(C=C2C1=O)C1=NC(NC2CCOCC2)=NC=C1Cl
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

molnova catalog
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