AM-6538

CAS No. 1245626-00-9

AM-6538 ( AM6538;AM 6538 )

Catalog No. M10994 CAS No. 1245626-00-9

AM-6538 (AM6538) is a potent, selective cannabinoid receptor CB1 antagonist with Ki of 5.1 nM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 336 Get Quote
50MG 1638 Get Quote
100MG 2250 Get Quote
200MG Get Quote Get Quote
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Biological Information

  • Product Name
    AM-6538
  • Note
    Research use only, not for human use.
  • Brief Description
    AM-6538 (AM6538) is a potent, selective cannabinoid receptor CB1 antagonist with Ki of 5.1 nM.
  • Description
    AM-6538 (AM6538) is a potent, selective cannabinoid receptor CB1 antagonist with Ki of 5.1 nM.
  • Synonyms
    AM6538;AM 6538
  • Pathway
    GPCR/G Protein
  • Target
    Cannabinoid Receptor
  • Recptor
    Cannabinoid Receptor
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1245626-00-9
  • Formula Weight
    542.42
  • Molecular Formula
    C26H25Cl2N5O4
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    O=[N+]([O-])OCCC#CC1=CC=C(C2=C(C)C(C(NN3CCCCC3)=O)=NN2C4=CC=C(Cl)C(Cl)=C4)C=C1
  • Chemical Name
    4-(4-(1-(2,4-dichlorophenyl)-4-methyl-3-(piperidin-1-ylcarbamoyl)-1H-pyrazol-5-yl)phenyl)but-3-yn-1-yl nitrate

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Hua T, et al. Cell. 2016 Oct 20;167(3):750-762.e14.
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