AM-2201
CAS No. 335161-24-5
AM-2201( AM 2201 | AM2201 )
Catalog No. M14138 CAS No. 335161-24-5
A synthetic cannabinoid that acts as a potent, nonselective full agonist for the cannabinoid receptor with EC50 of 38 and 58 nM for CB1 and CB2, respectively.
Purity : >98% (HPLC)
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100MG | Get Quote | In Stock |
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Biological Information
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Product NameAM-2201
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NoteResearch use only, not for human use.
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Brief DescriptionA synthetic cannabinoid that acts as a potent, nonselective full agonist for the cannabinoid receptor with EC50 of 38 and 58 nM for CB1 and CB2, respectively.
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DescriptionA synthetic cannabinoid that acts as a potent, nonselective full agonist for the cannabinoid receptor with EC50 of 38 and 58 nM for CB1 and CB2, respectively; dose-dependently induces hypothermia and reduces heart rate at doses of 0.3-10 mg/kg in mice.
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In Vitro——
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In Vivo——
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SynonymsAM 2201 | AM2201
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PathwayGPCR/G Protein
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TargetCannabinoid Receptor
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RecptorCannabinoid Receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number335161-24-5
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Formula Weight359.4
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Molecular FormulaC24H22FNO
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Purity>98% (HPLC)
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Solubility——
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SMILESc1ccc2c(c1)cccc2C(=O)c3cn(c4c3cccc4)CCCCCF
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Chemical Name[1-(5-fluoropentyl)-1H-indol-3-yl](naphthalene-1-yl)methanone
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
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Cannabichromene
Cannabichromene is a major non-psychotropic phytocannabinoid that inhibits endocannabinoid inactivation and activates the transient receptor potential ankyrin-1 (TRPA1).
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Hemopressin (rat)
Bioactive endogenous peptide substrate for endopeptidase 24.15 (ep24.15), neurolysin (ep24.16) and ACE. Ki values are 27.76, 3.43 and 1.87 μM respectively. Potent hypotensive in vivo. Also acts as a selective CB1 receptor inverse agonist. Displays antinociceptive activity and induces hypophagia in vivo.
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COR659
COR659 is a 2-acylaminothiophene derivative able to suppress alcohol and chocolate self-administration in rats, likely via positive allosteric modulation of the GABAB receptor and antagonism/inverse agonism at the cannabinoid CB1 receptor.