AF64394

CAS No. 1637300-25-4

AF64394 ( —— )

Catalog No. M21599 CAS No. 1637300-25-4

AF64394 is a selective inverse agonist of GPR3(pIC50 : 7.3).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 110 Get Quote
10MG 177 Get Quote
25MG 375 Get Quote
50MG 557 Get Quote
100MG 791 Get Quote
500MG 1611 Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    AF64394
  • Note
    Research use only not for human use.
  • Brief Description
    AF64394 is a selective inverse agonist of GPR3(pIC50 : 7.3).
  • Description
    AF64394 is a selective inverse agonist of GPR3(pIC50 : 7.3).
  • Synonyms
    ——
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    GPR3
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1637300-25-4
  • Formula Weight
    393.87
  • Molecular Formula
    C21H20ClN5O
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:125 mg/mL (317.36 mM)
  • SMILES
    CC(C)Oc1cc(Cl)ccc1CNc1cc(nc2ncnn12)-c1ccccc1
  • Chemical Name
    (4-Chloro-2-isopropoxy-benzyl)-(5-phenyl-[124]triazolo[15-a]pyrimidin-7-yl)-amine

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Jensen T et al. The identification of GPR3 inverse agonist AF64394; the first small molecule inhibitor of GPR3 receptor function. Bioorg Med Chem Lett. 2014 Nov 15;24(22):5195-8.
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