AF38469

CAS No. 1531634-31-7

AF38469( AF-38469 )

Catalog No. M23661 CAS No. 1531634-31-7

AF38469 is a new, specific and orally bioavailable Sortilin inhibitor (IC50: 330 nM).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 205 In Stock
10MG 335 In Stock
25MG 566 In Stock
50MG 806 In Stock
100MG 1098 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
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Biological Information

  • Product Name
    AF38469
  • Note
    Research use only, not for human use.
  • Brief Description
    AF38469 is a new, specific and orally bioavailable Sortilin inhibitor (IC50: 330 nM).
  • Description
    AF38469 is a new, specific and orally bioavailable Sortilin inhibitor (IC50: 330 nM).
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    AF-38469
  • Pathway
    GPCR/G Protein
  • Target
    Neurotensin Receptor
  • Recptor
    Sortilin
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1531634-31-7
  • Formula Weight
    324.25
  • Molecular Formula
    C15H11F3N2O3
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:40 mg/mL (123.36 mM)
  • SMILES
    Cc1cccc(NC(c(ccc(C(F)(F)F)c2)c2C(O)=O)=O)n1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Schroder TJ, et al. The identification of AF38469: an orally bioavailable inhibitor of the VPS10P family sorting receptor Sortilin. Bioorg Med Chem Lett. 2014 Jan 1;24(1):177-80.
molnova catalog
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