(S,R,S)-AHPC-C10-NH2

CAS No. 2341796-74-3

(S,R,S)-AHPC-C10-NH2 ( VH032-C10-NH2 )

Catalog No. M26943 CAS No. 2341796-74-3

(S,R,S)-AHPC-C10-NH2 is a synthesized E3 ligase ligand-linker conjugate incorporating the (S,R,S)-AHPC based VHL ligand and a linker used for BET-Targeted PROTAC.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 87 Get Quote
10MG 129 Get Quote
25MG 212 Get Quote
50MG 312 Get Quote
100MG 465 Get Quote
200MG Get Quote Get Quote
500MG Get Quote Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    (S,R,S)-AHPC-C10-NH2
  • Note
    Research use only, not for human use.
  • Brief Description
    (S,R,S)-AHPC-C10-NH2 is a synthesized E3 ligase ligand-linker conjugate incorporating the (S,R,S)-AHPC based VHL ligand and a linker used for BET-Targeted PROTAC.
  • Description
    (S,R,S)-AHPC-C10-NH2 is a synthesized E3 ligase ligand-linker conjugate incorporating the (S,R,S)-AHPC based VHL ligand and a linker used for BET-Targeted PROTAC.(In Vitro):PROTACs contain two different ligands connected by a linker; one is a ligand for an E3 ubiquitin ligase and the other is for the target protein. PROTACs exploit the intracellular ubiquitin-proteasome system to selectively degrade target proteins.
  • Synonyms
    VH032-C10-NH2
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    RGS19; RGS4
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2341796-74-3
  • Formula Weight
    613.9
  • Molecular Formula
    C33H51N5O4S
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCCCCN)C(C)(C)C)cc1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Levi L. Blazer et al.Reversible, Allosteric Small-Molecule Inhibitors of Regulator of G Protein Signaling Proteins. Molecular Pharmacology September 2010 vol.78 no.3 524-533
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