(S,R,S)-AHPC-C10-NH2
CAS No. 2341796-74-3
(S,R,S)-AHPC-C10-NH2 ( VH032-C10-NH2 )
Catalog No. M26943 CAS No. 2341796-74-3
(S,R,S)-AHPC-C10-NH2 is a synthesized E3 ligase ligand-linker conjugate incorporating the (S,R,S)-AHPC based VHL ligand and a linker used for BET-Targeted PROTAC.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
5MG | 87 | Get Quote |
|
10MG | 129 | Get Quote |
|
25MG | 212 | Get Quote |
|
50MG | 312 | Get Quote |
|
100MG | 465 | Get Quote |
|
200MG | Get Quote | Get Quote |
|
500MG | Get Quote | Get Quote |
|
1G | Get Quote | Get Quote |
|
Biological Information
-
Product Name(S,R,S)-AHPC-C10-NH2
-
NoteResearch use only, not for human use.
-
Brief Description(S,R,S)-AHPC-C10-NH2 is a synthesized E3 ligase ligand-linker conjugate incorporating the (S,R,S)-AHPC based VHL ligand and a linker used for BET-Targeted PROTAC.
-
Description(S,R,S)-AHPC-C10-NH2 is a synthesized E3 ligase ligand-linker conjugate incorporating the (S,R,S)-AHPC based VHL ligand and a linker used for BET-Targeted PROTAC.(In Vitro):PROTACs contain two different ligands connected by a linker; one is a ligand for an E3 ubiquitin ligase and the other is for the target protein. PROTACs exploit the intracellular ubiquitin-proteasome system to selectively degrade target proteins.
-
SynonymsVH032-C10-NH2
-
PathwayOthers
-
TargetOther Targets
-
RecptorRGS19; RGS4
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number2341796-74-3
-
Formula Weight613.9
-
Molecular FormulaC33H51N5O4S
-
Purity>98% (HPLC)
-
Solubility——
-
SMILESCc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCCCCN)C(C)(C)C)cc1
-
Chemical Name——
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1.Levi L. Blazer et al.Reversible, Allosteric Small-Molecule Inhibitors of Regulator of G Protein Signaling Proteins. Molecular Pharmacology September 2010 vol.78 no.3 524-533
molnova catalog
related products
-
Benfluorex hydrochlo...
Benfluorex is an anorectic and hypolipidemic agent that is structurally related to fenfluramine.
-
Tirzepatide hydrochl...
Tirzepatide hydrochloride (LY3298176 hydrochloride) is a dual glucose-dependent insulinotropic polypeptide (GIP) and glucagon-like peptide-1 (GLP-1) receptor agonist.
-
NGR peptide Trifluor...
NGR peptide Trifluoroacetate containing the asparagine-glycine-arginine (NGR) motif is recognized by CD13/aminopeptidase N (APN) receptor isoforms that are selectively overexpressed in tumor neovasculature.