(Rac)-AMG8379 ( (Rac)-AMG8380 )

Catalog No. M26409 CAS No. 1641574-26-6

(Rac)-AMG8379 is a racemate of AMG8379. AMG8379 is a potent, orally active and selective sulfonamide NaV1.7 antagonist(hNaV1.7 and mNaV1.7 with IC50s of 8.5 and 18.6 nM , respectively ).

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

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Size	Price / USD	Stock	Quantity
2MG	264	Get Quote
5MG	403	Get Quote
10MG	592	Get Quote
25MG	888	Get Quote
50MG	1242	Get Quote
100MG	1701	Get Quote
500MG	3402	Get Quote
1G	Get Quote	Get Quote

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Biological Information

Product Name

(Rac)-AMG8379
Note

Research use only, not for human use.
Brief Description

(Rac)-AMG8379 is a racemate of AMG8379. AMG8379 is a potent, orally active and selective sulfonamide NaV1.7 antagonist(hNaV1.7 and mNaV1.7 with IC50s of 8.5 and 18.6 nM , respectively ).
Description

(Rac)-AMG8379 is a racemate of AMG8379. AMG8379 is a potent, orally active and selective sulfonamide NaV1.7 antagonist(hNaV1.7 and mNaV1.7 with IC50s of 8.5 and 18.6 nM , respectively ).
Synonyms

(Rac)-AMG8380
Pathway

Others
Target

Other Targets
Recptor

ATF4; ATF6; ERK; GRP78; MMP
Research Area

——
Indication

——

Chemical Information

CAS Number

1641574-26-6
Formula Weight

543.9
Molecular Formula

C25H16ClF2N3O5S
Purity

>98% (HPLC)
Solubility

——
SMILES

O=S(NC1=NOC=C1)(C2=CC(C=CC(N3C4=CC(F)=C(C=C4OC)C5=CC(Cl)=CC(F)=C5)=O)=C3C=C2)=O.[Racemate]
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1.Zhang B, Han H, et al. Dehydroeffusol inhibits gastric cancer cell growth and tumorigenicity by selectively inducing tumor-suppressive endoplasmic reticulum stress and a moderate apoptosis. Biochem Pharmacol. 2016 Mar 15;104:8-18.

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