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(R)-Elagolix

CAS No. 834153-87-6

(R)-Elagolix ( NBI-56418 )

Catalog No. M24824 CAS No. 834153-87-6

(R)-Elagolix is a short-acting, nonpeptide, GnRH antagonist with an IC50 and Ki of 0.25 and 3.7 nM, respectively.?

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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5MG 65 In Stock
10MG 102 In Stock
25MG 178 In Stock
50MG 312 In Stock
100MG 462 In Stock
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Biological Information

  • Product Name
    (R)-Elagolix
  • Note
    Research use only, not for human use.
  • Brief Description
    (R)-Elagolix is a short-acting, nonpeptide, GnRH antagonist with an IC50 and Ki of 0.25 and 3.7 nM, respectively.?
  • Description
    (R)-Elagolix is a short-acting, nonpeptide, GnRH antagonist with an IC50 and Ki of 0.25 and 3.7 nM, respectively.?administered orally, that unlike injectable depot GnRH agonists and antagonists, produces a dose-dependent suppression of ovarian estrogen production, that is, from partial suppression at lower doses to full suppression at higher doses.
  • Synonyms
    NBI-56418
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    GnRHR
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    834153-87-6
  • Formula Weight
    631.6
  • Molecular Formula
    C32H30F5N3O5
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:100 mg/mL (158.33 mM)
  • SMILES
    CC1=C(C(=O)N(C(=O)N1CC2=C(C=CC=C2F)C(F)(F)F)C[C@@H](C3=CC=CC=C3)NCCCC(=O)O)C4=C(C(=CC=C4)OC)F
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Carr B, et al. Elagolix, an oral GnRH antagonist, versus subcutaneous depot medroxyprogesterone acetate for the treatment of endometriosis: effects on bone mineral density. Reprod Sci. 2014 Nov;21(11):1341-1351.
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