(R)-(-)-Rolipram
CAS No. 85416-75-7
(R)-(-)-Rolipram ( R)-Rolipram;(-)-Rolipram )
Catalog No. M16203 CAS No. 85416-75-7
A more active enantiomer of the PDE4 inhibitor rolipram.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
2MG | 35 | Get Quote |
|
5MG | 56 | Get Quote |
|
10MG | 88 | Get Quote |
|
25MG | 170 | Get Quote |
|
50MG | 317 | Get Quote |
|
100MG | Get Quote | Get Quote |
|
200MG | Get Quote | Get Quote |
|
500MG | Get Quote | Get Quote |
|
1G | Get Quote | Get Quote |
|
Biological Information
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Product Name(R)-(-)-Rolipram
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NoteResearch use only, not for human use.
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Brief DescriptionA more active enantiomer of the PDE4 inhibitor rolipram.
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DescriptionA more active enantiomer of the PDE4 inhibitor rolipram; shows 2-10-fold more potent than the S-(+) enantiomer rolipram.Asthma Phase 2 Clinical
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SynonymsR)-Rolipram;(-)-Rolipram
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PathwayAngiogenesis
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TargetPDE
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RecptorPDE
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Research AreaInflammation/Immunology
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IndicationAsthma
Chemical Information
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CAS Number85416-75-7
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Formula Weight275.34
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Molecular FormulaC16H21NO3
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Purity>98% (HPLC)
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SolubilityDMSO: ≥ 49 mg/mL
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SMILESCOC1=C(C=C(C=C1)C2CC(=O)NC2)OC3CCCC3
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Chemical Name2-Pyrrolidinone, 4-[3-(cyclopentyloxy)-4-methoxyphenyl]-, (4R)-
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Schneider HH, et al. Eur J Pharmacol. 1986 Aug 7;127(1-2):105-15.
2. Owens RJ, et al. Biochem J. 1997 Aug 15;326 ( Pt 1):53-60.
3. Ohsawa F, et al. Jpn J Pharmacol. 1998 Jun;77(2):147-54.
2. Owens RJ, et al. Biochem J. 1997 Aug 15;326 ( Pt 1):53-60.
3. Ohsawa F, et al. Jpn J Pharmacol. 1998 Jun;77(2):147-54.
molnova catalog
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