(E)-SI-2

Research use only, not for human use.

(E)-SI-2 is a potent small-molecule inhibitor of steroid receptor coactivator-3 (SRC-3 or AIB1) that can selectively inhibit the intrinsic transcriptional activities of SRC-3, also inhibits SRC-1 and SRC-2.

(E)-SI-2 is a potent small-molecule inhibitor of steroid receptor coactivator-3 (SRC-3 or AIB1) that can selectively inhibit the intrinsic transcriptional activities of SRC-3, also inhibits SRC-1 and SRC-2. It selectively reduces cellular protein levels of SRC-3, but not that of CARM-1, blocks MDA-MB-468 cell growth with an IC50 value of 3.4 nM, but spares normal cells.

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Others

Other Targets

Antibacterial

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380537-35-9

265.31

C15H15N5

>98% (HPLC)

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CN1C2=CC=CC=C2N=C1N/N=C(C3=NC=CC=C3)\C

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(-20℃)

With Ice Pack

≥ 2 years