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Ritanserin

CAS No. 87051-43-2

Ritanserin ( R 55667 )

Catalog No. M24881 CAS No. 87051-43-2

Ritanserin is a highly effective, relatively selective, long-acting antagonist of 5-HT2 receptor (IC50: 0.9 nM), less active on Histamine H1, Dopamine D2, Adrenergic α1, Adrenergic α2 receptors.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 43 In Stock
5MG 69 In Stock
10MG 104 In Stock
25MG 176 In Stock
50MG 259 In Stock
100MG 390 In Stock
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Biological Information

  • Product Name
    Ritanserin
  • Note
    Research use only, not for human use.
  • Brief Description
    Ritanserin is a highly effective, relatively selective, long-acting antagonist of 5-HT2 receptor (IC50: 0.9 nM), less active on Histamine H1, Dopamine D2, Adrenergic α1, Adrenergic α2 receptors.
  • Description
    Ritanserin is a highly effective, relatively selective, long-acting antagonist of 5-HT2 receptor (IC50: 0.9 nM), less active on Histamine H1, Dopamine D2, Adrenergic α1, Adrenergic α2 receptors.
  • Synonyms
    R 55667
  • Pathway
    Endocrinology/Hormones
  • Target
    5-HT Receptor
  • Recptor
    5-HT2;D2;H1 receptor;α1-adrenergic receptor;α2 receptor
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    87051-43-2
  • Formula Weight
    477.6
  • Molecular Formula
    C27H25F2N3OS
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:25 mg/mL (52.35 mM; Need ultrasonic)
  • SMILES
    CC1=C(C(N(C=CS2)C2=N1)=O)CCN(CC/3)CCC3=C(C4=CC=C(F)C=C4)\C5=CC=C(F)C=C5
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Leysen JE, et al. Receptor-binding properties in vitro and in vivo of ritanserin: A very potent and long acting serotonin-S2 antagonist. Mol Pharmacol. 1985 Jun;27(6):600-11.
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