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Ritanserin

CAS No. 87051-43-2

Ritanserin( R 55667 )

Catalog No. M24881 CAS No. 87051-43-2

Ritanserin is a highly effective, relatively selective, long-acting antagonist of 5-HT2 receptor (IC50: 0.9 nM), less active on Histamine H1, Dopamine D2, Adrenergic α1, Adrenergic α2 receptors.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 43 In Stock
5MG 69 In Stock
10MG 104 In Stock
25MG 176 In Stock
50MG 259 In Stock
100MG 390 In Stock
200MG Get Quote In Stock
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Biological Information

  • Product Name
    Ritanserin
  • Note
    Research use only, not for human use.
  • Brief Description
    Ritanserin is a highly effective, relatively selective, long-acting antagonist of 5-HT2 receptor (IC50: 0.9 nM), less active on Histamine H1, Dopamine D2, Adrenergic α1, Adrenergic α2 receptors.
  • Description
    Ritanserin is a highly effective, relatively selective, long-acting antagonist of 5-HT2 receptor (IC50: 0.9 nM), less active on Histamine H1, Dopamine D2, Adrenergic α1, Adrenergic α2 receptors.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    R 55667
  • Pathway
    Endocrinology/Hormones
  • Target
    5-HT Receptor
  • Recptor
    5-HT2|D2|H1 receptor|α1-adrenergic receptor|α2 receptor
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    87051-43-2
  • Formula Weight
    477.57
  • Molecular Formula
    C27H25F2N3OS
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:25 mg/mL (52.35 mM; Need ultrasonic)
  • SMILES
    CC1=C(C(N(C=CS2)C2=N1)=O)CCN(CC/3)CCC3=C(C4=CC=C(F)C=C4)\C5=CC=C(F)C=C5
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Leysen JE, et al. Receptor-binding properties in vitro and in vivo of ritanserin: A very potent and long acting serotonin-S2 antagonist. Mol Pharmacol. 1985 Jun;27(6):600-11.
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