Ritanserin ( R 55667 )

Catalog No. M24881 CAS No. 87051-43-2

Ritanserin is a highly effective, relatively selective, long-acting antagonist of 5-HT2 receptor (IC50: 0.9 nM), less active on Histamine H1, Dopamine D2, Adrenergic α1, Adrenergic α2 receptors.

Purity : >98% (HPLC)

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5MG	69	In Stock
10MG	104	In Stock
25MG	176	In Stock
50MG	259	In Stock
100MG	390	In Stock
200MG	Get Quote	In Stock
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Biological Information

Product Name

Ritanserin
Note

Research use only, not for human use.
Brief Description

Ritanserin is a highly effective, relatively selective, long-acting antagonist of 5-HT2 receptor (IC50: 0.9 nM), less active on Histamine H1, Dopamine D2, Adrenergic α1, Adrenergic α2 receptors.
Description

Ritanserin is a highly effective, relatively selective, long-acting antagonist of 5-HT2 receptor (IC50: 0.9 nM), less active on Histamine H1, Dopamine D2, Adrenergic α1, Adrenergic α2 receptors.
Synonyms

R 55667
Pathway

Endocrinology/Hormones
Target

5-HT Receptor
Recptor

5-HT2;D2;H1 receptor;α1-adrenergic receptor;α2 receptor
Research Area

——
Indication

——

Chemical Information

CAS Number

87051-43-2
Formula Weight

477.6
Molecular Formula

C27H25F2N3OS
Purity

>98% (HPLC)
Solubility

DMSO:25 mg/mL (52.35 mM; Need ultrasonic)
SMILES

CC1=C(C(N(C=CS2)C2=N1)=O)CCN(CC/3)CCC3=C(C4=CC=C(F)C=C4)\C5=CC=C(F)C=C5
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1.Leysen JE, et al. Receptor-binding properties in vitro and in vivo of ritanserin: A very potent and long acting serotonin-S2 antagonist. Mol Pharmacol. 1985 Jun;27(6):600-11.

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