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PNU-177864
CAS No. 250266-51-4
PNU-177864( —— )
Catalog No. M27686 CAS No. 250266-51-4
dopamine D3 receptor antagonist.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 132 | Get Quote |
|
| 5MG | 190 | Get Quote |
|
| 10MG | 237 | Get Quote |
|
| 25MG | 534 | Get Quote |
|
| 50MG | 762 | Get Quote |
|
| 100MG | 1053 | Get Quote |
|
| 500MG | 2097 | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NamePNU-177864
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NoteResearch use only, not for human use.
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Brief Descriptiondopamine D3 receptor antagonist.
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Descriptiondopamine D3 receptor antagonist.
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In Vitro——
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In VivoAnimal Model:Male and female Sprague-Dawley rats (8-9-week-old)Dosage:12.5 mg/kg, 50 mg/kg (for 2 weeks), or 200 mg/kg; 8 mg/kg, 25 mg/kg, or 80 mg/kg (for 4 weeks)Administration:Oral gavage; daily; for 2-4 weeksResult:Induced phospholipidosis in unusual target organs in dogs or rats including epididymis, pituitary, and hair follicles.
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Synonyms——
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PathwayOthers
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TargetOther Targets
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RecptorPI3K|Caspase|Bcl-2
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Research Area——
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Indication——
Chemical Information
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CAS Number250266-51-4
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Formula Weight438.89
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Molecular FormulaC18H21F3N2O3S·HCl
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Purity>98% (HPLC)
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Solubility——
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SMILESCCCNCCC1=CC=C(NS(C2=CC=C(OC(F)(F)F)C=C2)(=O)=O)C=C1.Cl
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Tomonaga T, et al. Isoflavonoids, genistein, psi-tectorigenin, and orobol, increase cytoplasmic free calcium in isolated rat hepatocytes. Biochem Biophys Res Commun. 1992 Jan 31;182(2):894-9.
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